Assay Detail
Binding
CHEMBL3135191
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Inhibition of human APT2
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Acyl protein thioesterase inhibitors as probes of dynamic S-palmitoylation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 7.11 | 7.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1903566 | — | — | 1 | 7.52 |
| CHEMBL3133033 | — | — | 1 | 6.70 |
| CHEMBL1891894 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1903566 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL3133033 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1891894 | — | IC50 | > | 10000.0 | nM | - |