Assay Detail
Binding
CHEMBL3214812
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Fluorescence-based biochemical high throughput screening dose response assay to identify inhibitors of Crimean-Congo Hemorrhagic Fever (CCHF) viral ovarian tumor domain protease (vOTU): Pep-AMC substrate. (Class of assay: confirmatory)
226
Total Activities
226
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 226 | 5.26 | 6.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1734083 | — | — | 1 | 6.89 |
| CHEMBL3189714 | — | — | 1 | 6.61 |
| CHEMBL1999630 | — | — | 1 | 6.59 |
| CHEMBL1598762 | — | — | 1 | 6.57 |
| CHEMBL1163377 | — | — | 1 | 6.56 |
| CHEMBL599924 | — | — | 1 | 6.56 |
| CHEMBL1384253 | — | — | 1 | 6.49 |
| CHEMBL1463659 | — | — | 1 | 6.44 |
| CHEMBL3191855 | — | — | 1 | 6.43 |
| CHEMBL1877709 | — | — | 1 | 6.42 |
| CHEMBL1728280 | — | — | 1 | 6.40 |
| CHEMBL2003651 | — | — | 1 | 6.40 |
| CHEMBL1210769 | — | — | 1 | 6.40 |
| CHEMBL3196451 | — | — | 1 | 6.39 |
| CHEMBL1735482 | — | — | 1 | 6.36 |
| CHEMBL339561 | — | — | 1 | 6.34 |
| CHEMBL3191689 | — | — | 1 | 6.15 |
| CHEMBL1335844 | — | — | 1 | 6.15 |
| CHEMBL1982305 | — | — | 1 | 6.11 |
| CHEMBL1546172 | — | — | 1 | 6.10 |
| CHEMBL3190880 | — | — | 1 | 6.08 |
| CHEMBL57013 | — | — | 1 | 6.03 |
| CHEMBL1721855 | — | — | 1 | 6.03 |
| CHEMBL1969046 | — | — | 1 | 6.01 |
| CHEMBL1453503 | — | — | 1 | 6.00 |
| CHEMBL1719244 | — | — | 1 | 5.98 |
| CHEMBL1471498 | — | — | 1 | 5.98 |
| CHEMBL1331912 | — | — | 1 | 5.95 |
| CHEMBL1505544 | — | — | 1 | 5.89 |
| CHEMBL1466516 | — | — | 1 | 5.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1734083 | — | IC50 | = | 127.24 | nM | 6.89 |
| CHEMBL3189714 | — | IC50 | = | 248.56 | nM | 6.61 |
| CHEMBL1999630 | — | IC50 | = | 256.73 | nM | 6.59 |
| CHEMBL1598762 | — | IC50 | = | 269.81 | nM | 6.57 |
| CHEMBL1163377 | — | IC50 | = | 275.83 | nM | 6.56 |
| CHEMBL599924 | — | IC50 | = | 275.73 | nM | 6.56 |
| CHEMBL1384253 | — | IC50 | = | 323.0 | nM | 6.49 |
| CHEMBL1463659 | — | IC50 | = | 366.21 | nM | 6.44 |
| CHEMBL3191855 | — | IC50 | = | 375.06 | nM | 6.43 |
| CHEMBL1877709 | — | IC50 | = | 384.4 | nM | 6.42 |
| CHEMBL1210769 | — | IC50 | = | 395.66 | nM | 6.40 |
| CHEMBL1728280 | — | IC50 | = | 396.15 | nM | 6.40 |
| CHEMBL2003651 | — | IC50 | = | 397.13 | nM | 6.40 |
| CHEMBL3196451 | — | IC50 | = | 405.13 | nM | 6.39 |
| CHEMBL1735482 | — | IC50 | = | 435.23 | nM | 6.36 |
| CHEMBL339561 | — | IC50 | = | 457.44 | nM | 6.34 |
| CHEMBL3191689 | — | IC50 | = | 701.35 | nM | 6.15 |
| CHEMBL1335844 | — | IC50 | = | 708.04 | nM | 6.15 |
| CHEMBL1982305 | — | IC50 | = | 771.17 | nM | 6.11 |
| CHEMBL1546172 | — | IC50 | = | 786.51 | nM | 6.10 |
| CHEMBL3190880 | — | IC50 | = | 833.09 | nM | 6.08 |
| CHEMBL1721855 | — | IC50 | = | 945.0 | nM | 6.03 |
| CHEMBL57013 | — | IC50 | = | 931.0 | nM | 6.03 |
| CHEMBL1969046 | — | IC50 | = | 973.0 | nM | 6.01 |
| CHEMBL1453503 | — | IC50 | = | 1003.0 | nM | 6.00 |
| CHEMBL1719244 | — | IC50 | = | 1046.0 | nM | 5.98 |
| CHEMBL1471498 | — | IC50 | = | 1053.0 | nM | 5.98 |
| CHEMBL1331912 | — | IC50 | = | 1135.0 | nM | 5.95 |
| CHEMBL1505544 | — | IC50 | = | 1282.0 | nM | 5.89 |
| CHEMBL1466516 | — | IC50 | = | 1280.0 | nM | 5.89 |
| CHEMBL1359236 | — | IC50 | = | 1342.0 | nM | 5.87 |
| CHEMBL1702473 | — | IC50 | = | 1372.0 | nM | 5.86 |
| CHEMBL284328 | HOMIDIUM BROMIDE | IC50 | = | 1558.0 | nM | 5.81 |
| CHEMBL1964407 | — | IC50 | = | 1574.0 | nM | 5.80 |
| CHEMBL3197091 | — | IC50 | = | 1720.0 | nM | 5.76 |
| CHEMBL1713009 | — | IC50 | = | 1776.0 | nM | 5.75 |
| CHEMBL171632 | — | IC50 | = | 1835.0 | nM | 5.74 |
| CHEMBL1706454 | — | IC50 | = | 1870.0 | nM | 5.73 |
| CHEMBL156174 | — | IC50 | = | 1855.0 | nM | 5.73 |
| CHEMBL1698802 | — | IC50 | = | 1935.0 | nM | 5.71 |
| CHEMBL429095 | — | IC50 | = | 2150.0 | nM | 5.67 |
| CHEMBL1733422 | — | IC50 | = | 2163.0 | nM | 5.67 |
| CHEMBL1452795 | — | IC50 | = | 2353.0 | nM | 5.63 |
| CHEMBL51931 | 9,10-PHENANTHRENEQUINONE | IC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL1329974 | — | IC50 | = | 2444.0 | nM | 5.61 |
| CHEMBL1542693 | — | IC50 | = | 2433.0 | nM | 5.61 |
| CHEMBL1709883 | — | IC50 | = | 2503.0 | nM | 5.60 |
| CHEMBL3216654 | — | IC50 | = | 2521.0 | nM | 5.60 |
| CHEMBL1732365 | — | IC50 | = | 2511.0 | nM | 5.60 |
| CHEMBL2141749 | — | IC50 | = | 2560.0 | nM | 5.59 |