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Assay Detail

CHEMBL3224328

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimalarial activity against chloroquine-sensitive Plasmodium falciparum
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Antimalarial peroxides: advances in drug discovery and design
Slack RD, Jacobine AM, Posner GH
Medchemcomm (2012) 3 : 281 -297
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 10 8.36 8.41

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3221639 1 8.41
CHEMBL3221880 1 8.41
CHEMBL3221879 1 8.41
CHEMBL3221878 1 8.41
CHEMBL3221877 1 8.41
CHEMBL3221876 1 8.41
CHEMBL3221875 1 8.41
CHEMBL269513 1 8.40
CHEMBL3221873 1 8.15
CHEMBL3221874 1 8.15

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3221639 IC50 = 3.9 nM 8.41
CHEMBL3221880 IC50 = 3.9 nM 8.41
CHEMBL3221879 IC50 = 3.9 nM 8.41
CHEMBL3221878 IC50 = 3.9 nM 8.41
CHEMBL3221877 IC50 = 3.9 nM 8.41
CHEMBL3221876 IC50 = 3.9 nM 8.41
CHEMBL3221875 IC50 = 3.9 nM 8.41
CHEMBL269513 IC50 = 4.0 nM 8.40
CHEMBL3221873 IC50 = 7.0 nM 8.15
CHEMBL3221874 IC50 = 7.0 nM 8.15