Assay Detail
Binding
CHEMBL3225244
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Binding affinity to human recombinant MAOA
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Identification of multifunctional small molecule-based reversible monoamine oxidase inhibitors
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 7 | 5.70 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3219618 | — | — | 1 | 7.00 |
| CHEMBL3219619 | — | — | 1 | 6.72 |
| CHEMBL1984524 | — | — | 1 | 5.64 |
| CHEMBL3219620 | — | — | 1 | 5.60 |
| CHEMBL3219621 | — | — | 1 | 5.29 |
| CHEMBL402456 | — | — | 1 | 5.24 |
| CHEMBL3219617 | — | — | 1 | 4.43 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3219618 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL3219619 | — | Ki | = | 190.0 | nM | 6.72 |
| CHEMBL1984524 | — | Ki | = | 2300.0 | nM | 5.64 |
| CHEMBL3219620 | — | Ki | = | 2500.0 | nM | 5.60 |
| CHEMBL3219621 | — | Ki | = | 5100.0 | nM | 5.29 |
| CHEMBL402456 | — | Ki | = | 5700.0 | nM | 5.24 |
| CHEMBL3219617 | — | Ki | = | 37000.0 | nM | 4.43 |