Assay Detail
Binding
CHEMBL3227237
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Binding affinity to adenosine A3 receptor (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Methanocarba ring as a ribose modification in ligands of G protein-coupled purine and pyrimidine receptors: synthetic approaches.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 7.24 | 8.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL27809 | — | — | 1 | 8.66 |
| CHEMBL417292 | — | — | 1 | 8.39 |
| CHEMBL308634 | — | — | 1 | 4.66 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL27809 | — | Ki | = | 2.2 | nM | 8.66 |
| CHEMBL417292 | — | Ki | = | 4.1 | nM | 8.39 |
| CHEMBL308634 | — | Ki | = | 22000.0 | nM | 4.66 |