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Assay Detail

CHEMBL3238920

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]SR141716A from rat CB1 receptor expressed in CHO-K1 cells by liquid scintillation spectrophotometry
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Cell Type CHO-K1
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cannabinoid receptor 1 (CHEMBL3571)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Therapeutic utility of cannabinoid receptor type 2 (CB(2)) selective agonists.
Han S, Thatte J, Buzard DJ, Jones RM.
J Med Chem (2013) 56 : 8224 -8256
PubMed 23865723 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.59 5.59

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL495528 1 5.59

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL495528 Ki = 2565.0 nM 5.59