Assay Detail
Binding
CHEMBL3238923
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Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO-K1 cells by liquid scintillation counting
6
Total Activities
6
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO-K1 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Therapeutic utility of cannabinoid receptor type 2 (CB(2)) selective agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 6.08 | 6.57 |
| EC50 | 3 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1668519 | — | — | 1 | 6.57 |
| CHEMBL3234708 | — | — | 1 | 5.58 |
| CHEMBL495528 | — | — | 1 | - |
| CHEMBL3234698 | — | — | 1 | - |
| CHEMBL3234699 | — | — | 1 | - |
| CHEMBL3235055 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1668519 | — | Ki | = | 272.0 | nM | 6.57 |
| CHEMBL3234708 | — | Ki | = | 2630.0 | nM | 5.58 |
| CHEMBL495528 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL3234698 | — | EC50 | > | 27000.0 | nM | - |
| CHEMBL3234699 | — | EC50 | > | 27000.0 | nM | - |
| CHEMBL3235055 | — | EC50 | > | 50000.0 | nM | - |