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Assay Detail

CHEMBL3240176

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Growth inhibition of HUVEC by WST-8 assay
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HUVEC
Confidence 1 — Organism
Curated By Autocuration

Target

HUVEC (CHEMBL613979)
Type CELL-LINE
Organism Homo sapiens

Publication

Potential anti-angiogenesis effects of p-terphenyl compounds from Polyozellus multiplex.
Nagasawa I, Kaneko A, Suzuki T, Nishio K, Kinoshita K, Shiro M, Koyama K.
J Nat Prod (2014) 77 : 963 -968
PubMed 24601669 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 5.22 5.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL178455 1 5.85
CHEMBL3236668 1 5.47
CHEMBL3236669 1 5.12
CHEMBL458248 POLYOZELLIN 1 4.99
CHEMBL3236670 1 4.67

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL178455 IC50 = 1400.0 nM 5.85
CHEMBL3236668 IC50 = 3400.0 nM 5.47
CHEMBL3236669 IC50 = 7600.0 nM 5.12
CHEMBL458248 POLYOZELLIN IC50 = 10200.0 nM 4.99
CHEMBL3236670 IC50 = 21400.0 nM 4.67