Assay Detail
Binding
CHEMBL3240237
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of metallo-beta-lactamase VIM2 (unknown origin)
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Not specified |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
The applications of binuclear metallohydrolases in medicine: recent advances in the design and development of novel drug leads for purple acid phosphatases, metallo-β-lactamases and arginases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 5.82 | 5.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3234718 | — | — | 1 | 5.82 |
| CHEMBL3234719 | — | — | 1 | 5.82 |
| CHEMBL3234720 | — | — | 1 | 5.82 |
| CHEMBL3234721 | — | — | 1 | 5.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3234718 | — | Ki | = | 1500.0 | nM | 5.82 |
| CHEMBL3234719 | — | Ki | = | 1500.0 | nM | 5.82 |
| CHEMBL3234720 | — | Ki | = | 1500.0 | nM | 5.82 |
| CHEMBL3234721 | — | Ki | = | 1500.0 | nM | 5.82 |