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Assay Detail

CHEMBL3243108

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of DNP-BSA-stimulated TNF-alpha production in rat RBL2H3 cells preincubated for 15 mins followed by DNP-BSA addition measured after 3 hrs by ELISA
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Rattus norvegicus
Cell Type RBL-2H3
Confidence 1 — Organism
Curated By Autocuration

Target

RBL-2H3 (CHEMBL614632)
Type CELL-LINE
Organism Rattus norvegicus

Publication

Structural elucidation and synthesis of vialinin C, a new inhibitor of TNF-α production.
Ye YQ, Negishi C, Hongo Y, Koshino H, Onose J, Abe N, Takahashi S.
Bioorg Med Chem (2014) 22 : 2442 -2446
PubMed 24679673 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 10.05 10.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2012938 VIALININ A 1 10.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2012938 VIALININ A IC50 = 0.09 nM 10.05