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Assay Detail

CHEMBL3257007

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of porcine pancreatic kallikrein
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Sus scrofa
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Glandular kallikrein (CHEMBL3243909)
Type SINGLE PROTEIN
Organism Sus scrofa

Publication

Structure-activity relationships for the inhibition of acrosin by benzamidine derivatives.
Parrish RF, Straus JW, Paulson JD, Polakoski KL, Tidwell RR, Geratz JD, Stevens FM.
J Med Chem (1978) 21 : 1132 -1136
PubMed 722718 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.41 7.41

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3245418 1 7.41

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3245418 Ki = 39.3 nM 7.41