Assay Detail
Binding
CHEMBL3292179
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of IKKbeta kinase (unknown origin) by Lance ULight system
23
Total Activities
23
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Inhibitor of nuclear factor kappa-B kinase subunit beta (CHEMBL1991) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Discovery of thienopyrimidine-based FLT3 inhibitors from the structural modification of known IKKβ inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 23 | 7.21 | 7.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL129857 | AS-602868 | 1.0 | 1 | 7.21 |
| CHEMBL3290618 | — | — | 1 | - |
| CHEMBL3290634 | — | — | 1 | - |
| CHEMBL3290632 | — | — | 1 | - |
| CHEMBL3290631 | — | — | 1 | - |
| CHEMBL3290630 | — | — | 1 | - |
| CHEMBL3290629 | — | — | 1 | - |
| CHEMBL3290624 | — | — | 1 | - |
| CHEMBL3290623 | — | — | 1 | - |
| CHEMBL3290622 | — | — | 1 | - |
| CHEMBL3290621 | — | — | 1 | - |
| CHEMBL3290620 | — | — | 1 | - |
| CHEMBL3290613 | — | — | 1 | - |
| CHEMBL3290617 | — | — | 1 | - |
| CHEMBL3290616 | — | — | 1 | - |
| CHEMBL3290615 | — | — | 1 | - |
| CHEMBL3290614 | — | — | 1 | - |
| CHEMBL3290625 | — | — | 1 | - |
| CHEMBL3290626 | — | — | 1 | - |
| CHEMBL3290627 | — | — | 1 | - |
| CHEMBL3290628 | — | — | 1 | - |
| CHEMBL3290633 | — | — | 1 | - |
| CHEMBL3290619 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL129857 | AS-602868 | IC50 | = | 62.0 | nM | 7.21 |
| CHEMBL3290618 | — | IC50 | - | — | - | |
| CHEMBL3290634 | — | IC50 | - | — | - | |
| CHEMBL3290632 | — | IC50 | - | — | - | |
| CHEMBL3290631 | — | IC50 | - | — | - | |
| CHEMBL3290630 | — | IC50 | - | — | - | |
| CHEMBL3290629 | — | IC50 | - | — | - | |
| CHEMBL3290624 | — | IC50 | - | — | - | |
| CHEMBL3290623 | — | IC50 | - | — | - | |
| CHEMBL3290622 | — | IC50 | - | — | - | |
| CHEMBL3290621 | — | IC50 | - | — | - | |
| CHEMBL3290620 | — | IC50 | - | — | - | |
| CHEMBL3290613 | — | IC50 | - | — | - | |
| CHEMBL3290617 | — | IC50 | - | — | - | |
| CHEMBL3290616 | — | IC50 | - | — | - | |
| CHEMBL3290615 | — | IC50 | - | — | - | |
| CHEMBL3290614 | — | IC50 | - | — | - | |
| CHEMBL3290625 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3290626 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3290627 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3290628 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3290633 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3290619 | — | IC50 | - | — | - |