Assay Detail
Binding
CHEMBL3295084
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]WAY-100635 from 5-HT1A receptor in pig cerebral cortex homogenates by competitive binding assay
21
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Sus scrofa |
| Tissue | Cerebral cortex |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Functionally selective dopamine D₂, D₃ receptor partial agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 21 | 7.48 | 9.31 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2028019 | CARIPRAZINE | 4.0 | 1 | 9.31 |
| CHEMBL3287403 | — | — | 2 | 8.38 |
| CHEMBL3287396 | — | — | 1 | 8.24 |
| CHEMBL3287404 | — | — | 1 | 8.15 |
| CHEMBL3287399 | — | — | 1 | 7.82 |
| CHEMBL3287406 | — | — | 1 | 7.80 |
| CHEMBL3287394 | — | — | 1 | 7.77 |
| CHEMBL3287401 | — | — | 1 | 7.54 |
| CHEMBL3287400 | — | — | 1 | 7.51 |
| CHEMBL3287402 | — | — | 1 | 7.44 |
| CHEMBL3287398 | — | — | 1 | 7.38 |
| CHEMBL3287393 | — | — | 1 | 7.37 |
| CHEMBL3287395 | — | — | 1 | 7.32 |
| CHEMBL3287392 | — | — | 1 | 7.09 |
| CHEMBL3287391 | — | — | 1 | 7.08 |
| CHEMBL1112 | ARIPIPRAZOLE | 4.0 | 1 | 7.06 |
| CHEMBL3287397 | — | — | 1 | 7.02 |
| CHEMBL3287405 | — | — | 1 | 7.01 |
| CHEMBL3287390 | — | — | 1 | 6.96 |
| CHEMBL240773 | QUINPIROLE | 2.0 | 1 | 5.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2028019 | CARIPRAZINE | Ki | = | 0.49 | nM | 9.31 |
| CHEMBL3287403 | — | Ki | = | 4.2 | nM | 8.38 |
| CHEMBL3287396 | — | Ki | = | 5.7 | nM | 8.24 |
| CHEMBL3287404 | — | Ki | = | 7.1 | nM | 8.15 |
| CHEMBL3287399 | — | Ki | = | 15.0 | nM | 7.82 |
| CHEMBL3287406 | — | Ki | = | 16.0 | nM | 7.80 |
| CHEMBL3287394 | — | Ki | = | 17.0 | nM | 7.77 |
| CHEMBL3287403 | — | Ki | = | 21.0 | nM | 7.68 |
| CHEMBL3287401 | — | Ki | = | 29.0 | nM | 7.54 |
| CHEMBL3287400 | — | Ki | = | 31.0 | nM | 7.51 |
| CHEMBL3287402 | — | Ki | = | 36.0 | nM | 7.44 |
| CHEMBL3287398 | — | Ki | = | 42.0 | nM | 7.38 |
| CHEMBL3287393 | — | Ki | = | 43.0 | nM | 7.37 |
| CHEMBL3287395 | — | Ki | = | 48.0 | nM | 7.32 |
| CHEMBL3287392 | — | Ki | = | 82.0 | nM | 7.09 |
| CHEMBL3287391 | — | Ki | = | 83.0 | nM | 7.08 |
| CHEMBL1112 | ARIPIPRAZOLE | Ki | = | 88.0 | nM | 7.06 |
| CHEMBL3287397 | — | Ki | = | 95.0 | nM | 7.02 |
| CHEMBL3287405 | — | Ki | = | 98.0 | nM | 7.01 |
| CHEMBL3287390 | — | Ki | = | 110.0 | nM | 6.96 |
| CHEMBL240773 | QUINPIROLE | Ki | = | 6300.0 | nM | 5.20 |