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Assay Detail

CHEMBL3296168

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against human HEK293T cells assessed as cell viability after 48 hrs by MTT assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type HEK-293T
Confidence 1 — Organism
Curated By Autocuration

Target

HEK-293T (CHEMBL3706568)
Type CELL-LINE
Organism Homo sapiens

Publication

Dithiaarsanes induce oxidative stress-mediated apoptosis in HL-60 cells by selectively targeting thioredoxin reductase.
Liu Y, Duan D, Yao J, Zhang B, Peng S, Ma H, Song Y, Fang J.
J Med Chem (2014) 57 : 5203 -5211
PubMed 24867309 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.57 5.57

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3290761 1 5.57

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3290761 IC50 = 2700.0 nM 5.57