Assay Detail
Functional
CHEMBL3296830
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Anticancer against human HT-29 cells assessed as cell viability after 48 hrs by SRB assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HT-29 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Bismuth nitrate-induced novel nitration of estradiol: an entry to new anticancer agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 6 | 5.39 | 6.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3287935 | — | — | 1 | 6.77 |
| CHEMBL3287936 | — | — | 1 | 5.50 |
| CHEMBL3287934 | — | — | 1 | 5.37 |
| CHEMBL1627573 | — | — | 1 | 5.21 |
| CHEMBL3287933 | — | — | 1 | 4.96 |
| CHEMBL1627935 | — | — | 1 | 4.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3287935 | — | IC50 | = | 170.0 | nM | 6.77 |
| CHEMBL3287936 | — | IC50 | = | 3200.0 | nM | 5.50 |
| CHEMBL3287934 | — | IC50 | = | 4300.0 | nM | 5.37 |
| CHEMBL1627573 | — | IC50 | = | 6200.0 | nM | 5.21 |
| CHEMBL3287933 | — | IC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL1627935 | — | IC50 | = | 28800.0 | nM | 4.54 |