Assay Detail
Functional
CHEMBL3362622
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human NMUR2 expressed in CHO cells by calcium mobilization assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of selective hexapeptide agonists to human neuromedin U receptors types 1 and 2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 8.40 | 8.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3315349 | — | — | 1 | 8.60 |
| CHEMBL3315335 | — | — | 1 | 8.19 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3315349 | — | EC50 | = | 2.5 | nM | 8.60 |
| CHEMBL3315335 | — | EC50 | = | 6.4 | nM | 8.19 |