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Assay Detail

CHEMBL3364246

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhbition of Influenza A virus (A/X-31(H3N2) hemagglutinin binding to 2 hrs compound pre-incubated MDCK cells assessed as reduction in viral RNA measured after 1 hr by RT-qPCR analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Influenza A virus (A/X-31(H3N2))
Cell Type MDCK
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Semisynthetic teicoplanin derivatives as new influenza virus binding inhibitors: synthesis and antiviral studies.
Bereczki I, Kicsák M, Dobray L, Borbás A, Batta G, Kéki S, Nikodém ÉN, Ostorházi E, Rozgonyi F, Vanderlinden E, Naesens L, Herczegh P.
Bioorg Med Chem Lett (2014) 24 : 3251 -3254
PubMed 24974341 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.25 5.33

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3310642 1 5.33
CHEMBL3310643 1 5.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3310642 IC50 = 4700.0 nM 5.33
CHEMBL3310643 IC50 = 7000.0 nM 5.16