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Assay Detail

CHEMBL3364447

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of mushroom tyrosinase using L-DOPA as substrate by spectrophotometry relative to control
5
Total Activities
3
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Agaricus bisporus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Tyrosinase (CHEMBL3318)
Type SINGLE PROTEIN
Organism Agaricus bisporus

Publication

Effect of p-aminophenols on tyrosinase activity.
Komori Y, Imai M, Yamauchi T, Higashiyama K, Takahashi N.
Bioorg Med Chem (2014) 22 : 3994 -4000
PubMed 24972725 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 4.50 4.52
Inhibition 2 - -

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL427462 2 4.52
CHEMBL287556 KOJIC ACID 1 4.48
CHEMBL376316 2 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL427462 IC50 = 30100.0 nM 4.52
CHEMBL287556 KOJIC ACID IC50 = 32800.0 nM 4.48
CHEMBL376316 IC50 > 200000.0 nM -
CHEMBL376316 Inhibition - % -
CHEMBL427462 Inhibition - % -