Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL3364757

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Physicochemical
Antioxidant activity assessed as DPPH radical scavenging capacity after 30 mins by UV spectrophotometry
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Physicochemical
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Publication

Antioxidant effects of the highly-substituted carbazole alkaloids and their related carbazoles.
Hieda Y, Anraku M, Choshi T, Tomida H, Fujioka H, Hatae N, Hori O, Hirose J, Hibino S.
Bioorg Med Chem Lett (2014) 24 : 3530 -3533
PubMed 24928405 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 11 4.98 5.21

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL7983 PROPYL GALLATE 1.0 1 5.21
CHEMBL3309627 1 5.15
CHEMBL3309629 1 5.12
CHEMBL3309628 1 5.01
CHEMBL3309626 1 5.00
CHEMBL3309632 1 4.92
CHEMBL3309631 1 4.92
CHEMBL3309625 1 4.92
CHEMBL47 ALPHA-TOCOPHEROL 1 4.81
CHEMBL290916 EDARAVONE 4.0 1 4.71
CHEMBL3309630 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL7983 PROPYL GALLATE IC50 = 6100.0 nM 5.21
CHEMBL3309627 IC50 = 7100.0 nM 5.15
CHEMBL3309629 IC50 = 7600.0 nM 5.12
CHEMBL3309628 IC50 = 9800.0 nM 5.01
CHEMBL3309626 IC50 = 9900.0 nM 5.00
CHEMBL3309632 IC50 = 12000.0 nM 4.92
CHEMBL3309631 IC50 = 12000.0 nM 4.92
CHEMBL3309625 IC50 = 12000.0 nM 4.92
CHEMBL47 ALPHA-TOCOPHEROL IC50 = 15400.0 nM 4.81
CHEMBL290916 EDARAVONE IC50 = 19700.0 nM 4.71
CHEMBL3309630 IC50 > 50000.0 nM -