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Assay Detail

CHEMBL3364758

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Physicochemical
Antioxidant activity assessed as ABTS+ radical scavenging capacity after 16 hrs by UV spectrophotometry
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Physicochemical
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Publication

Antioxidant effects of the highly-substituted carbazole alkaloids and their related carbazoles.
Hieda Y, Anraku M, Choshi T, Tomida H, Fujioka H, Hatae N, Hori O, Hirose J, Hibino S.
Bioorg Med Chem Lett (2014) 24 : 3530 -3533
PubMed 24928405 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 11 4.26 4.28

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3309627 1 4.28
CHEMBL3309629 1 4.24
CHEMBL3309632 1 -
CHEMBL3309631 1 -
CHEMBL3309630 1 -
CHEMBL3309628 1 -
CHEMBL3309626 1 -
CHEMBL3309625 1 -
CHEMBL290916 EDARAVONE 4.0 1 -
CHEMBL47 ALPHA-TOCOPHEROL 1 -
CHEMBL7983 PROPYL GALLATE 1.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3309627 IC50 = 52600.0 nM 4.28
CHEMBL3309629 IC50 = 57100.0 nM 4.24
CHEMBL3309632 IC50 = 174600.0 nM -
CHEMBL3309631 IC50 = 160600.0 nM -
CHEMBL3309630 IC50 > 500000.0 nM -
CHEMBL3309628 IC50 = 115900.0 nM -
CHEMBL3309626 IC50 = 111700.0 nM -
CHEMBL3309625 IC50 = 158900.0 nM -
CHEMBL290916 EDARAVONE IC50 = 213700.0 nM -
CHEMBL47 ALPHA-TOCOPHEROL IC50 = 211100.0 nM -
CHEMBL7983 PROPYL GALLATE IC50 = 187500.0 nM -