Assay Detail
Binding
CHEMBL3367270
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of xanthine oxidase (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Flavones: an important scaffold for medicinal chemistry.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 5.65 | 6.28 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL28 | APIGENIN | — | 1 | 6.28 |
| CHEMBL151 | LUTEOLIN | 2.0 | 1 | 5.54 |
| CHEMBL1467 | ALLOPURINOL | 4.0 | 1 | 5.14 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL28 | APIGENIN | Ki | = | 520.0 | nM | 6.28 |
| CHEMBL151 | LUTEOLIN | Ki | = | 2900.0 | nM | 5.54 |
| CHEMBL1467 | ALLOPURINOL | Ki | = | 7300.0 | nM | 5.14 |