Assay Detail
Functional
CHEMBL3367910
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Antiplasmodial activity against Plasmodium falciparum 3D7
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Plasmodium falciparum |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Target evaluation of deoxyhypusine synthase from Theileria parva the neglected animal parasite and its relationship to Plasmodium.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 6.80 | 7.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL587083 | — | — | 1 | 7.08 |
| CHEMBL532879 | — | — | 1 | 6.85 |
| CHEMBL547488 | — | — | 1 | 6.46 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL587083 | — | EC50 | = | 82.2 | nM | 7.08 |
| CHEMBL532879 | — | EC50 | = | 142.0 | nM | 6.85 |
| CHEMBL547488 | — | EC50 | = | 345.0 | nM | 6.46 |