Assay Detail
Binding
CHEMBL3368016
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Nav1.7 (unknown origin) by PatchXpress method
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Sodium channel protein type 9 subunit alpha (CHEMBL4296) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Recent progress in sodium channel modulators for pain.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 8.77 | 9.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3341983 | — | — | 1 | 9.22 |
| CHEMBL3341984 | — | — | 1 | 8.68 |
| CHEMBL3341985 | — | — | 1 | 8.42 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3341983 | — | IC50 | = | 0.6 | nM | 9.22 |
| CHEMBL3341984 | — | IC50 | = | 2.1 | nM | 8.68 |
| CHEMBL3341985 | — | IC50 | = | 3.8 | nM | 8.42 |