Assay Detail
Binding
CHEMBL3385406
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to SUR1 (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
ATP-binding cassette sub-family C member 8 (CHEMBL2071) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Novel sulfonyl(thio)urea derivatives act efficiently both as insulin secretagogues and as insulinomimetic compounds.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 9.05 | 9.42 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3330880 | — | — | 1 | 9.42 |
| CHEMBL3330879 | — | — | 1 | 8.68 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3330880 | — | Kd | = | 0.38 | nM | 9.42 |
| CHEMBL3330879 | — | Kd | = | 2.08 | nM | 8.68 |