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Assay Detail

CHEMBL3386565

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimicrobial activity against multidrug-resistant Plasmodium falciparum FCR3 assessed as growth inhibition after 3 days by HRP2-based ELISA
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Binding modes of reverse fosmidomycin analogs toward the antimalarial target IspC.
Konzuch S, Umeda T, Held J, Hähn S, Brücher K, Lienau C, Behrendt CT, Gräwert T, Bacher A, Illarionov B, Fischer M, Mordmüller B, Tanaka N, Kurz T.
J Med Chem (2014) 57 : 8827 -8838
PubMed 25254502 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 6.35 6.42

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2164256 1 6.42
CHEMBL3342262 1 6.39
CHEMBL3341763 1 6.24

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2164256 IC50 = 380.0 nM 6.42
CHEMBL3342262 IC50 = 410.0 nM 6.39
CHEMBL3341763 IC50 = 570.0 nM 6.24