Assay Detail
Binding
CHEMBL3390778
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of STAT5B SH2 domain (unknown origin)-5-FAM-GpYLVLDKW interaction compound treated for 15 mins by fluorescent polarization assay
25
Total Activities
25
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Signal transducer and activator of transcription 5B (CHEMBL5817) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Nanomolar-Potency Small Molecule Inhibitor of STAT5 Protein.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 25 | 5.44 | 6.84 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3358611 | — | — | 1 | 6.84 |
| CHEMBL3358598 | — | — | 1 | 5.32 |
| CHEMBL3358596 | — | — | 1 | 5.18 |
| CHEMBL3358610 | — | — | 1 | 4.94 |
| CHEMBL3358608 | — | — | 1 | 4.91 |
| CHEMBL3358609 | — | — | 1 | - |
| CHEMBL3358607 | — | — | 1 | - |
| CHEMBL3358606 | — | — | 1 | - |
| CHEMBL3358605 | — | — | 1 | - |
| CHEMBL3358604 | — | — | 1 | - |
| CHEMBL3358603 | — | — | 1 | - |
| CHEMBL3358602 | — | — | 1 | - |
| CHEMBL3358601 | — | — | 1 | - |
| CHEMBL3358600 | — | — | 1 | - |
| CHEMBL3358599 | — | — | 1 | - |
| CHEMBL3358597 | — | — | 1 | - |
| CHEMBL3358595 | — | — | 1 | - |
| CHEMBL3358594 | — | — | 1 | - |
| CHEMBL3358593 | — | — | 1 | - |
| CHEMBL3358592 | — | — | 1 | - |
| CHEMBL3358591 | — | — | 1 | - |
| CHEMBL3358590 | — | — | 1 | - |
| CHEMBL3358589 | — | — | 1 | - |
| CHEMBL3358588 | — | — | 1 | - |
| CHEMBL3358587 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3358611 | — | Ki | = | 145.8 | nM | 6.84 |
| CHEMBL3358598 | — | Ki | = | 4770.0 | nM | 5.32 |
| CHEMBL3358596 | — | Ki | = | 6620.0 | nM | 5.18 |
| CHEMBL3358610 | — | Ki | = | 11500.0 | nM | 4.94 |
| CHEMBL3358608 | — | Ki | = | 12360.0 | nM | 4.91 |
| CHEMBL3358609 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358607 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358606 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358605 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358604 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358603 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358602 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358601 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358600 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358599 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358597 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358595 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358594 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358593 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358592 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358591 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358590 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358589 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358588 | — | Ki | > | 60000.0 | nM | - |
| CHEMBL3358587 | — | Ki | > | 60000.0 | nM | - |