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Assay Detail

CHEMBL3391509

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of p300 (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Histone acetyltransferase p300 (CHEMBL3784)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Development of second generation epigenetic agents
Jones P
Medchemcomm (2012) 3 : 135 -161
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.72 7.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL505121 1 7.72

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL505121 Ki = 19.0 nM 7.72