Assay Detail
Binding
CHEMBL3394985
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Activation of human AMPK alpha1beta1gamma1
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Target
AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1 (CHEMBL2111345) ↗| Type | PROTEIN COMPLEX |
| Organism | Homo sapiens |
Publication
Small molecule adenosine 5'-monophosphate activated protein kinase (AMPK) modulators and human diseases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 10 | 8.08 | 9.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3393129 | — | — | 1 | 9.22 |
| CHEMBL3393128 | — | — | 1 | 9.00 |
| CHEMBL3393130 | — | — | 1 | 8.96 |
| CHEMBL3393127 | — | — | 1 | 8.52 |
| CHEMBL3393131 | — | — | 1 | 8.40 |
| CHEMBL3393133 | — | — | 1 | 7.89 |
| CHEMBL3393132 | — | — | 1 | 7.77 |
| CHEMBL3393136 | — | — | 1 | 7.24 |
| CHEMBL3393134 | — | — | 1 | 7.01 |
| CHEMBL3393135 | — | — | 1 | 6.74 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3393129 | — | EC50 | = | 0.6 | nM | 9.22 |
| CHEMBL3393128 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3393130 | — | EC50 | = | 1.1 | nM | 8.96 |
| CHEMBL3393127 | — | EC50 | = | 3.0 | nM | 8.52 |
| CHEMBL3393131 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3393133 | — | EC50 | = | 13.0 | nM | 7.89 |
| CHEMBL3393132 | — | EC50 | = | 17.0 | nM | 7.77 |
| CHEMBL3393136 | — | EC50 | = | 58.0 | nM | 7.24 |
| CHEMBL3393134 | — | EC50 | = | 97.0 | nM | 7.01 |
| CHEMBL3393135 | — | EC50 | = | 184.0 | nM | 6.74 |