Assay Detail
Functional
CHEMBL3398868
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human recombinant DP1 receptor by cAMP assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of a new series of potent prostacyclin receptor agonists with in vivo activity in rat.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 6.63 | 6.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3398236 | — | — | 1 | 6.85 |
| CHEMBL3398228 | — | — | 1 | 6.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3398236 | — | EC50 | = | 140.0 | nM | 6.85 |
| CHEMBL3398228 | — | EC50 | = | 400.0 | nM | 6.40 |