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Assay Detail

CHEMBL3399752

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Binding
Inhibition of HCV genotype 3a NS5B RNA dependent RNA polymerase assessed as reduction in triphosphate activity
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Hepatitis C virus subtype 3a
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Synthesis and characterization of 1'-C-cyano-2'-fluoro-2'-C-methyl pyrimidine nucleosides as HCV polymerase inhibitors.
Kirschberg TA, Mish MR, Zhang L, Squires NH, Wang KY, Cho A, Feng JY, Fenaux M, Babusis D, Park Y, Ray AS, Kim CU.
Bioorg Med Chem Lett (2015) 25 : 1040 -1043
PubMed 25650256 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.16 6.16

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL510394 1 6.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL510394 IC50 = 700.0 nM 6.16