Assay Detail
Binding
CHEMBL3404599
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]LSD from human cloned 5-HT6R expressed in HEK293 cells using seven compounds concentrations
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Fingerprint-based consensus virtual screening towards structurally new 5-HT(6)R ligands.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.55 | 6.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1580288 | — | — | 1 | 6.92 |
| CHEMBL2011865 | — | — | 1 | 6.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1580288 | — | Ki | = | 119.0 | nM | 6.92 |
| CHEMBL2011865 | — | Ki | = | 670.0 | nM | 6.17 |