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Assay Detail

CHEMBL3411100

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Antagonist activity at human NK1 receptor expressed in CHO cells by luminescence assay in presence of SP peptide
16
Total Activities
16
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type CHO
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Substance-P receptor (CHEMBL249)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist - neurokinin-1 antagonist peptidomimetics.
Guillemyn K, Kleczkowska P, Lesniak A, Dyniewicz J, Van der Poorten O, Van den Eynde I, Keresztes A, Varga E, Lai J, Porreca F, Chung NN, Lemieux C, Mika J, Rojewska E, Makuch W, Van Duppen J, Przewlocka B, Vanden Broeck J, Lipkowski AW, Schiller PW, Tourwé D, Ballet S.
Eur J Med Chem (2015) 92 : 64 -77
PubMed 25544687 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
pA2 11 - -
Kd 5 6.99 8.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1782139 1 8.40
CHEMBL1782141 1 7.80
CHEMBL3408519 1 6.44
CHEMBL3408520 1 6.27
CHEMBL3408518 1 6.04
CHEMBL3408737 1 -
CHEMBL3408736 1 -
CHEMBL3408735 1 -
CHEMBL3408734 1 -
CHEMBL3408733 1 -
CHEMBL3408732 1 -
CHEMBL3408731 1 -
CHEMBL3408730 1 -
CHEMBL3408522 1 -
CHEMBL3408521 1 -
CHEMBL1782140 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1782139 Kd = 3.981 nM 8.40
CHEMBL1782141 Kd = 15.85 nM 7.80
CHEMBL3408519 Kd = 363.08 nM 6.44
CHEMBL3408520 Kd = 537.03 nM 6.27
CHEMBL3408518 Kd = 912.01 nM 6.04
CHEMBL3408737 pA2 - -
CHEMBL3408736 pA2 - -
CHEMBL3408735 pA2 - -
CHEMBL3408734 pA2 - -
CHEMBL3408733 pA2 - -
CHEMBL3408732 pA2 - -
CHEMBL3408731 pA2 - -
CHEMBL3408730 pA2 - -
CHEMBL3408522 pA2 - -
CHEMBL3408521 pA2 - -
CHEMBL1782140 pA2 - -