Assay Detail
Functional
CHEMBL3412052
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Anticancer activity against human TALL-1 cells assessed as cell number by coulter channelyzer
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | TALL-1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
BMS-871: a novel orally active pan-Notch inhibitor as an anticancer agent.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 14 | 8.08 | 8.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3410151 | — | — | 1 | 8.52 |
| CHEMBL3410161 | — | — | 1 | 8.40 |
| CHEMBL3410166 | — | — | 1 | 8.40 |
| CHEMBL3410168 | — | — | 1 | 8.40 |
| CHEMBL3410169 | — | — | 1 | 8.40 |
| CHEMBL3410170 | — | — | 1 | 8.40 |
| CHEMBL3410167 | — | — | 1 | 8.30 |
| CHEMBL3410163 | — | — | 1 | 7.89 |
| CHEMBL3410162 | — | — | 1 | 7.82 |
| CHEMBL3410164 | — | — | 1 | 7.58 |
| CHEMBL3410154 | — | — | 1 | 6.80 |
| CHEMBL3410152 | — | — | 1 | - |
| CHEMBL3410153 | — | — | 1 | - |
| CHEMBL3410165 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3410151 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL3410161 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3410166 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3410168 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3410169 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3410170 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3410167 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL3410163 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL3410162 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL3410164 | — | IC50 | = | 26.0 | nM | 7.58 |
| CHEMBL3410154 | — | IC50 | = | 158.0 | nM | 6.80 |
| CHEMBL3410152 | — | IC50 | - | — | - | |
| CHEMBL3410153 | — | IC50 | - | — | - | |
| CHEMBL3410165 | — | IC50 | - | — | - |