Assay Detail
Binding
CHEMBL3418797
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Inhibition of CK2 (unknown origin)
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Identification of protein kinase CK2 inhibitors using solvent dipole ordering virtual screening.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 6 | 6.11 | 7.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1231683 | — | — | 1 | 7.52 |
| CHEMBL92361 | — | — | 1 | 6.41 |
| CHEMBL28 | APIGENIN | — | 1 | 6.10 |
| CHEMBL177820 | TETRABROMOBENZOTRIAZOLE | — | 1 | 6.05 |
| CHEMBL289277 | EMODIN | — | 1 | 5.70 |
| CHEMBL3706697 | — | — | 1 | 4.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1231683 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL92361 | — | IC50 | = | 390.0 | nM | 6.41 |
| CHEMBL28 | APIGENIN | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL177820 | TETRABROMOBENZOTRIAZOLE | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL289277 | EMODIN | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL3706697 | — | IC50 | = | 13000.0 | nM | 4.89 |