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Assay Detail

CHEMBL3424239

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Growth inhibition of mouse B16 cells by MTT method
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type B16
Confidence 1 — Organism
Curated By Autocuration

Target

B16 (CHEMBL381)
Type CELL-LINE
Organism Mus musculus

Publication

1,19-seco-Avermectin analogues from a ΔaveCDE mutant Streptomyces avermectinius strain.
Sun P, Zhao Q, Wu Z, Zhang W, Liu W.
J Nat Prod (2015) 78 : 301 -305
PubMed 25611131 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 4.71 5.19

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL359744 DOXORUBICIN HYDROCHLORIDE 4.0 1 5.19
CHEMBL3422422 1 4.83
CHEMBL1630577 ABAMECTIN COMPONENT B1A -1.0 1 4.69
CHEMBL3422424 1 4.46
CHEMBL3422423 1 4.39

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL359744 DOXORUBICIN HYDROCHLORIDE IC50 = 6400.0 nM 5.19
CHEMBL3422422 IC50 = 14700.0 nM 4.83
CHEMBL1630577 ABAMECTIN COMPONENT B1A IC50 = 20500.0 nM 4.69
CHEMBL3422424 IC50 = 35100.0 nM 4.46
CHEMBL3422423 IC50 = 40600.0 nM 4.39