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Assay Detail

CHEMBL3428359

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human CD38 extracellular domain expressed in Pichia pastoris assessed as NAD hydrolysis by colorimetric-based assay
84
Total Activities
84
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1 (CHEMBL4660)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery, Synthesis, and Biological Evaluation of Thiazoloquin(az)olin(on)es as Potent CD38 Inhibitors.
Haffner CD, Becherer JD, Boros EE, Cadilla R, Carpenter T, Cowan D, Deaton DN, Guo Y, Harrington W, Henke BR, Jeune MR, Kaldor I, Milliken N, Petrov KG, Preugschat F, Schulte C, Shearer BG, Shearer T, Smalley TL, Stewart EL, Stuart JD, Ulrich JC.
J Med Chem (2015) 58 : 3548 -3571
PubMed 25828863 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 84 6.51 8.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3426065 1 8.85
CHEMBL3426064 1 8.47
CHEMBL3426037 1 8.42
CHEMBL3426033 1 8.41
CHEMBL3426066 1 8.32
CHEMBL3426067 1 8.28
CHEMBL3426032 1 8.22
CHEMBL3426034 1 8.14
CHEMBL3426035 1 8.00
CHEMBL3426038 1 7.89
CHEMBL3426040 1 7.85
CHEMBL3426039 1 7.82
CHEMBL3426058 1 7.58
CHEMBL3426057 1 7.55
CHEMBL3426061 1 7.38
CHEMBL3426188 1 7.31
CHEMBL3426063 1 7.30
CHEMBL3426060 1 7.28
CHEMBL3426031 1 7.28
CHEMBL3426036 1 7.27
CHEMBL3426029 1 7.26
CHEMBL3426027 1 7.24
CHEMBL3426028 1 7.21
CHEMBL3426059 1 7.19
CHEMBL3426191 1 7.11
CHEMBL3426030 1 7.05
CHEMBL3426193 1 7.04
CHEMBL3426186 1 6.93
CHEMBL3426094 1 6.88
CHEMBL3426187 1 6.85

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3426065 IC50 = 1.4 nM 8.85
CHEMBL3426064 IC50 = 3.4 nM 8.47
CHEMBL3426037 IC50 = 3.8 nM 8.42
CHEMBL3426033 IC50 = 3.9 nM 8.41
CHEMBL3426066 IC50 = 4.8 nM 8.32
CHEMBL3426067 IC50 = 5.3 nM 8.28
CHEMBL3426032 IC50 = 6.0 nM 8.22
CHEMBL3426034 IC50 = 7.3 nM 8.14
CHEMBL3426035 IC50 = 10.0 nM 8.00
CHEMBL3426038 IC50 = 13.0 nM 7.89
CHEMBL3426040 IC50 = 14.0 nM 7.85
CHEMBL3426039 IC50 = 15.0 nM 7.82
CHEMBL3426058 IC50 = 26.0 nM 7.58
CHEMBL3426057 IC50 = 28.0 nM 7.55
CHEMBL3426061 IC50 = 42.0 nM 7.38
CHEMBL3426188 IC50 = 49.0 nM 7.31
CHEMBL3426063 IC50 = 50.0 nM 7.30
CHEMBL3426060 IC50 = 53.0 nM 7.28
CHEMBL3426031 IC50 = 52.0 nM 7.28
CHEMBL3426036 IC50 = 54.0 nM 7.27
CHEMBL3426029 IC50 = 55.0 nM 7.26
CHEMBL3426027 IC50 = 58.0 nM 7.24
CHEMBL3426028 IC50 = 61.0 nM 7.21
CHEMBL3426059 IC50 = 64.0 nM 7.19
CHEMBL3426191 IC50 = 78.0 nM 7.11
CHEMBL3426030 IC50 = 89.0 nM 7.05
CHEMBL3426193 IC50 = 92.0 nM 7.04
CHEMBL3426186 IC50 = 117.0 nM 6.93
CHEMBL3426094 IC50 = 132.0 nM 6.88
CHEMBL3426187 IC50 = 140.0 nM 6.85
CHEMBL3426189 IC50 = 142.0 nM 6.85
CHEMBL3426184 IC50 = 149.0 nM 6.83
CHEMBL3426056 IC50 = 206.0 nM 6.69
CHEMBL3426062 IC50 = 245.0 nM 6.61
CHEMBL3426055 IC50 = 263.0 nM 6.58
CHEMBL3426093 IC50 = 281.0 nM 6.55
CHEMBL3426068 IC50 = 298.0 nM 6.53
CHEMBL3426190 IC50 = 406.0 nM 6.39
CHEMBL3426086 IC50 = 460.0 nM 6.34
CHEMBL3426043 IC50 = 498.0 nM 6.30
CHEMBL3426084 IC50 = 560.0 nM 6.25
CHEMBL3426081 IC50 = 700.0 nM 6.16
CHEMBL3426072 IC50 = 700.0 nM 6.16
CHEMBL3426085 IC50 = 840.0 nM 6.08
CHEMBL3426069 IC50 = 840.0 nM 6.08
CHEMBL3426090 IC50 = 950.0 nM 6.02
CHEMBL3426044 IC50 = 959.0 nM 6.02
CHEMBL3426082 IC50 = 970.0 nM 6.01
CHEMBL3426192 IC50 = 971.0 nM 6.01
CHEMBL3426075 IC50 = 970.0 nM 6.01