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Assay Detail

CHEMBL3562040

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PubChem BioAssay. Luminescence-based cell-based high throughput dose response assay to identify inhibitors of viability of late stage Plasmodium falciparum gametocytes. (Class of assay: confirmatory)
244
Total Activities
244
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category confirmatory
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 244 4.77 5.07

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1488923 1 5.07
CHEMBL1526953 1 5.04
CHEMBL1612044 1 4.82
CHEMBL1327810 1 4.54
CHEMBL1310318 1 4.40
CHEMBL1735080 1 -
CHEMBL1896411 1 -
CHEMBL1577914 1 -
CHEMBL1409255 1 -
CHEMBL1611089 1 -
CHEMBL1608285 1 -
CHEMBL1510756 1 -
CHEMBL1579514 1 -
CHEMBL1577160 1 -
CHEMBL1422167 1 -
CHEMBL1536198 1 -
CHEMBL1399835 1 -
CHEMBL1341808 1 -
CHEMBL1901165 1 -
CHEMBL1390245 1 -
CHEMBL2141346 1 -
CHEMBL1471955 1 -
CHEMBL1374100 1 -
CHEMBL1450241 1 -
CHEMBL1450769 1 -
CHEMBL1306159 1 -
CHEMBL1371320 1 -
CHEMBL1392521 1 -
CHEMBL1499751 1 -
CHEMBL1299736 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1488923 IC50 = 8597.0 nM 5.07
CHEMBL1526953 IC50 = 9125.0 nM 5.04
CHEMBL1612044 IC50 = 15244.0 nM 4.82
CHEMBL1327810 IC50 = 28818.0 nM 4.54
CHEMBL1310318 IC50 = 39617.0 nM 4.40
CHEMBL1537115 IC50 > 108787.0 nM -
CHEMBL1511162 IC50 > 108791.0 nM -
CHEMBL1488986 IC50 > 108814.0 nM -
CHEMBL1306513 IC50 > 108787.0 nM -
CHEMBL1557251 IC50 > 108787.0 nM -
CHEMBL1711210 IC50 > 108803.0 nM -
CHEMBL1563978 IC50 > 108814.0 nM -
CHEMBL1611227 IC50 > 108786.0 nM -
CHEMBL1385485 IC50 > 108723.0 nM -
CHEMBL2132231 IC50 > 108836.0 nM -
CHEMBL1309203 IC50 > 108797.0 nM -
CHEMBL1550466 IC50 > 108789.0 nM -
CHEMBL1540629 IC50 > 108790.0 nM -
CHEMBL1385373 IC50 > 108793.0 nM -
CHEMBL1302969 IC50 > 108803.0 nM -
CHEMBL1454182 IC50 > 108779.0 nM -
CHEMBL1423114 IC50 > 108890.0 nM -
CHEMBL1438544 IC50 > 108923.0 nM -
CHEMBL1584386 IC50 > 108724.0 nM -
CHEMBL1537854 IC50 > 108803.0 nM -
CHEMBL1599872 IC50 > 108825.0 nM -
CHEMBL1386428 IC50 > 108814.0 nM -
CHEMBL1509711 IC50 > 108716.0 nM -
CHEMBL1372869 IC50 > 108814.0 nM -
CHEMBL1582830 IC50 > 108858.0 nM -
CHEMBL1497135 IC50 > 108796.0 nM -
CHEMBL1429875 IC50 > 108803.0 nM -
CHEMBL1377718 IC50 > 108792.0 nM -
CHEMBL1483420 IC50 > 108802.0 nM -
CHEMBL1402896 IC50 > 108638.0 nM -
CHEMBL1428728 IC50 > 108814.0 nM -
CHEMBL1448921 IC50 > 108763.0 nM -
CHEMBL1732171 IC50 > 108847.0 nM -
CHEMBL1904115 IC50 > 108825.0 nM -
CHEMBL1891973 IC50 > 108814.0 nM -
CHEMBL1351569 IC50 > 108766.0 nM -
CHEMBL1477713 IC50 > 108803.0 nM -
CHEMBL1335486 IC50 > 108732.0 nM -
CHEMBL1426363 IC50 > 108879.0 nM -
CHEMBL1705197 IC50 > 108814.0 nM -
CHEMBL1369541 IC50 > 108724.0 nM -
CHEMBL1402652 IC50 > 108836.0 nM -
CHEMBL1390959 IC50 > 108890.0 nM -
CHEMBL3561308 IC50 > 108765.0 nM -
CHEMBL1611944 IC50 > 108814.0 nM -