Assay Detail
Functional
CHEMBL3580214
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Anticancer activity against human MDA-MB-231 cells assessed as cell growth inhibition after 20 to 70 hrs by Real-time RTCA iCELLgence system
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MDA-MB-231 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Studies on the ATP Binding Site of Fyn Kinase for the Identification of New Inhibitors and Their Evaluation as Potential Agents against Tauopathies and Tumors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.26 | 5.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3578214 | — | — | 1 | 5.43 |
| CHEMBL3578215 | — | — | 1 | 5.08 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3578214 | — | IC50 | = | 3700.0 | nM | 5.43 |
| CHEMBL3578215 | — | IC50 | = | 8300.0 | nM | 5.08 |