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Assay Detail

CHEMBL3584374

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against wild type Hepatitis B virus
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepatitis B virus
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis B virus (CHEMBL613497)
Type ORGANISM
Organism Hepatitis B virus

Publication

Synthesis and biological evaluation of 4-substituted fluoronucleoside analogs for the treatment of hepatitis B virus infection.
Yang Q, Kang J, Zheng L, Wang XJ, Wan N, Wu J, Qiao Y, Niu P, Wang SQ, Peng Y, Wang Q, Yu W, Chang J.
J Med Chem (2015) 58 : 3693 -3703
PubMed 25905540 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 6.92 6.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL519846 RO-0622 3.0 1 6.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL519846 RO-0622 EC50 = 120.0 nM 6.92