Assay Detail
Binding
CHEMBL3591679
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Inhibition of JHDM1F (unknown origin) using H3K9mel peptide
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Identification of Jumonji AT-Rich Interactive Domain 1A Inhibitors and Their Effect on Cancer Cells.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 17 | 4.39 | 4.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3590431 | — | — | 1 | 4.62 |
| CHEMBL3590430 | — | — | 1 | 4.54 |
| CHEMBL3590421 | — | — | 1 | 4.24 |
| CHEMBL3590427 | — | — | 1 | 4.14 |
| CHEMBL3590418 | — | — | 1 | - |
| CHEMBL3590419 | — | — | 1 | - |
| CHEMBL3590420 | — | — | 1 | - |
| CHEMBL3590422 | — | — | 1 | - |
| CHEMBL3590423 | — | — | 1 | - |
| CHEMBL3590424 | — | — | 1 | - |
| CHEMBL90852 | N-OXALYLGLYCINE | — | 1 | - |
| CHEMBL3590426 | — | — | 1 | - |
| CHEMBL3590428 | — | — | 1 | - |
| CHEMBL3590429 | — | — | 1 | - |
| CHEMBL3590432 | — | — | 1 | - |
| CHEMBL3590433 | — | — | 1 | - |
| CHEMBL3590425 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3590431 | — | IC50 | = | 24000.0 | nM | 4.62 |
| CHEMBL3590430 | — | IC50 | = | 29000.0 | nM | 4.54 |
| CHEMBL3590421 | — | IC50 | = | 58000.0 | nM | 4.24 |
| CHEMBL3590427 | — | IC50 | = | 73000.0 | nM | 4.14 |
| CHEMBL3590418 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3590419 | — | IC50 | - | — | - | |
| CHEMBL3590420 | — | IC50 | - | — | - | |
| CHEMBL3590422 | — | IC50 | - | — | - | |
| CHEMBL3590423 | — | IC50 | - | — | - | |
| CHEMBL3590424 | — | IC50 | - | — | - | |
| CHEMBL90852 | N-OXALYLGLYCINE | IC50 | = | 640000.0 | nM | - |
| CHEMBL3590426 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3590428 | — | IC50 | - | — | - | |
| CHEMBL3590429 | — | IC50 | - | — | - | |
| CHEMBL3590432 | — | IC50 | - | — | - | |
| CHEMBL3590433 | — | IC50 | - | — | - | |
| CHEMBL3590425 | — | IC50 | - | — | - |