Assay Detail
Binding
CHEMBL3598449
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of ST6N (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Beta-galactoside alpha-2,6-sialyltransferase 1 (CHEMBL3596075) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Beyond substrate analogues: new inhibitor chemotypes for glycosyltransferases
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.35 | 6.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1170899 | — | — | 1 | 6.21 |
| CHEMBL1170697 | — | — | 1 | 5.10 |
| CHEMBL3596263 | — | — | 1 | 4.73 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1170899 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL1170697 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL3596263 | — | IC50 | = | 18500.0 | nM | 4.73 |