Assay Detail
Binding
CHEMBL3598455
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of rat ST6Gal1
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Beta-galactoside alpha-2,6-sialyltransferase 1 (CHEMBL4276) ↗| Type | SINGLE PROTEIN |
| Organism | Rattus norvegicus |
Publication
Beyond substrate analogues: new inhibitor chemotypes for glycosyltransferases
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.51 | 5.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL122701 | — | — | 1 | 5.72 |
| CHEMBL222556 | — | — | 1 | 5.29 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL122701 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL222556 | — | IC50 | = | 5100.0 | nM | 5.29 |