Assay Detail
Physicochemical
CHEMBL3602222
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Inhibition of beta-hematin formation
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Physicochemical |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
From hybrid compounds to targeted drug delivery in antimalarial therapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.25 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1096247 | — | — | 1 | 8.70 |
| CHEMBL1254709 | DM-1157 | 1.0 | 1 | 5.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1096247 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL1254709 | DM-1157 | IC50 | = | 1600.0 | nM | 5.80 |