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Assay Detail

CHEMBL3602223

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Functional
Antimalarial activity against Plasmodium falciparum NF54 assessed as inhibition of parasite growth
3
Total Activities
3
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

From hybrid compounds to targeted drug delivery in antimalarial therapy.
Oliveira R, Miranda D, Magalhães J, Capela R, Perry MJ, O'Neill PM, Moreira R, Lopes F.
Bioorg Med Chem (2015) 23 : 5120 -5130
PubMed 25913864 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
MIC 2 - -
IC50 1 8.15 8.15

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1096247 1 8.15
CHEMBL76 CHLOROQUINE 4.0 1 -
CHEMBL1289388 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1096247 IC50 = 7.1 nM 8.15
CHEMBL76 CHLOROQUINE MIC = 0.125 ug.mL-1 -
CHEMBL1289388 MIC = 0.25 ug.mL-1 -