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Assay Detail

CHEMBL3602688

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Binding
Inhibition of Influenza A/PR/8/34 (H1N1) core RNA-dependent RNA polymerase endonuclease activity using cap1 alfalfa mosaic virus RNA as substrate after 60 mins by liquid scintillation counting analysis in presence of [35S]-UTP
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Influenza A virus (A/Puerto Rico/8/1934(H1N1))
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Structural and computational study on inhibitory compounds for endonuclease activity of influenza virus polymerase.
Fudo S, Yamamoto N, Nukaga M, Odagiri T, Tashiro M, Neya S, Hoshino T.
Bioorg Med Chem (2015) 23 : 5466 -5475
PubMed 26252962 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.37 6.37

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL463590 1 6.37

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL463590 IC50 = 430.0 nM 6.37