Assay Detail
Functional
CHEMBL3603632
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Growth inhibition of human HT-29 cells after 72 hrs by APH assay
16
Total Activities
16
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HT-29 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Design, Synthesis, and Biological Evaluation of a Series of Anthracene-9,10-dione Dioxime β-Catenin Pathway Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| GI50 | 15 | - | - |
| IC50 | 1 | 6.70 | 6.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3601410 | — | — | 1 | 6.70 |
| CHEMBL3601411 | TEGAVIVINT | 2.0 | 1 | - |
| CHEMBL3601480 | — | — | 1 | - |
| CHEMBL3601481 | — | — | 1 | - |
| CHEMBL3601482 | — | — | 1 | - |
| CHEMBL3601483 | — | — | 1 | - |
| CHEMBL3601484 | — | — | 1 | - |
| CHEMBL3601485 | — | — | 1 | - |
| CHEMBL3601486 | — | — | 1 | - |
| CHEMBL3601487 | — | — | 1 | - |
| CHEMBL3601488 | — | — | 1 | - |
| CHEMBL3601489 | — | — | 1 | - |
| CHEMBL3601490 | — | — | 1 | - |
| CHEMBL3601491 | — | — | 1 | - |
| CHEMBL3601492 | — | — | 1 | - |
| CHEMBL3601493 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3601410 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL3601411 | TEGAVIVINT | GI50 | = | 90.0 | nM | - |
| CHEMBL3601480 | — | GI50 | = | 600.0 | nM | - |
| CHEMBL3601481 | — | GI50 | = | 190.0 | nM | - |
| CHEMBL3601482 | — | GI50 | = | 140.0 | nM | - |
| CHEMBL3601483 | — | GI50 | = | 30.0 | nM | - |
| CHEMBL3601484 | — | GI50 | = | 20.0 | nM | - |
| CHEMBL3601485 | — | GI50 | = | 80.0 | nM | - |
| CHEMBL3601486 | — | GI50 | = | 470.0 | nM | - |
| CHEMBL3601487 | — | GI50 | = | 60.0 | nM | - |
| CHEMBL3601488 | — | GI50 | = | 90.0 | nM | - |
| CHEMBL3601489 | — | GI50 | > | 100000.0 | nM | - |
| CHEMBL3601490 | — | GI50 | = | 60.0 | nM | - |
| CHEMBL3601491 | — | GI50 | = | 180.0 | nM | - |
| CHEMBL3601492 | — | GI50 | = | 80.0 | nM | - |
| CHEMBL3601493 | — | GI50 | = | 3900.0 | nM | - |