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Assay Detail

CHEMBL3607084

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HCMV infected in HFF after 3 days by neutral red dye-based plaque reduction assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human betaherpesvirus 5
Confidence 1 — Organism
Curated By Autocuration

Target

Human betaherpesvirus 5 (CHEMBL371)
Type ORGANISM
Organism Human betaherpesvirus 5

Publication

2- and 3-Fluoro-3-deazaneplanocins, 2-fluoro-3-deazaaristeromycins, and 3-methyl-3-deazaneplanocin: Synthesis and antiviral properties.
Liu C, Chen Q, Gorden JD, Schneller SW.
Bioorg Med Chem (2015) 23 : 5496 -5501
PubMed 26260336 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 5.50 6.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3604361 1 6.52
CHEMBL182 GANCICLOVIR 4.0 1 5.44
CHEMBL3604362 1 5.29
CHEMBL3603846 1 5.19
CHEMBL3604363 1 5.06
CHEMBL3604364 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3604361 IC50 = 300.0 nM 6.52
CHEMBL182 GANCICLOVIR IC50 = 3600.0 nM 5.44
CHEMBL3604362 IC50 = 5100.0 nM 5.29
CHEMBL3603846 IC50 = 6400.0 nM 5.19
CHEMBL3604363 IC50 = 8700.0 nM 5.06
CHEMBL3604364 IC50 < 100.0 nM -