Assay Detail
Binding
CHEMBL3618944
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of mouse NaV1.6 channel by two-electrode voltage-clamp method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Sodium channel protein type 8 subunit alpha (CHEMBL1914275) ↗| Type | SINGLE PROTEIN |
| Organism | Mus musculus |
Publication
Voltage-Gated Sodium Channels: Structure, Function, Pharmacology, and Clinical Indications.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.62 | 6.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3617066 | — | — | 1 | 6.62 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3617066 | — | IC50 | = | 240.0 | nM | 6.62 |