Assay Detail
Functional
CHEMBL3620199
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Cytotoxicity against human HeLa cells by MTT assay
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HeLa |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Cytotoxic cardenolides from the latex of Calotropis procera.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 10 | 6.36 | 7.06 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3617462 | — | — | 1 | 7.06 |
| CHEMBL3617460 | — | — | 1 | 6.98 |
| CHEMBL3617459 | — | — | 1 | 6.89 |
| CHEMBL500585 | USCHARIN | — | 1 | 6.56 |
| CHEMBL3617463 | — | — | 1 | 6.50 |
| CHEMBL3617461 | — | — | 1 | 6.18 |
| CHEMBL522203 | — | — | 1 | 6.06 |
| CHEMBL3617464 | — | — | 1 | 5.94 |
| CHEMBL3617465 | — | — | 1 | 5.84 |
| CHEMBL3617466 | — | — | 1 | 5.61 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3617462 | — | IC50 | = | 87.0 | nM | 7.06 |
| CHEMBL3617460 | — | IC50 | = | 104.0 | nM | 6.98 |
| CHEMBL3617459 | — | IC50 | = | 128.0 | nM | 6.89 |
| CHEMBL500585 | USCHARIN | IC50 | = | 275.0 | nM | 6.56 |
| CHEMBL3617463 | — | IC50 | = | 318.0 | nM | 6.50 |
| CHEMBL3617461 | — | IC50 | = | 663.0 | nM | 6.18 |
| CHEMBL522203 | — | IC50 | = | 863.0 | nM | 6.06 |
| CHEMBL3617464 | — | IC50 | = | 1151.0 | nM | 5.94 |
| CHEMBL3617465 | — | IC50 | = | 1434.0 | nM | 5.84 |
| CHEMBL3617466 | — | IC50 | = | 2472.0 | nM | 5.61 |