Assay Detail
Binding
CHEMBL3624254
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [32P]diazirine-LPA from LPA receptor in mouse N1E-115 cells preincubated for 1 hr in dark followed by UV irradiation for 5 mins by scintillation counting analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Cell Type | N1E-115 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
The status of the lysophosphatidic acid receptor type 1 (LPA1R)
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 8.00 | 8.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL117021 | LYSOPHOSPHATIDIC ACID | — | 1 | 8.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL117021 | LYSOPHOSPHATIDIC ACID | IC50 | = | 10.0 | nM | 8.00 |